SCHEMBL364256

SCHEMBL364256

Cc1ccccc1C(CC(=O)c1c[nH]c(=O)c(C)c1)c1ccc(C(=O)NC[C@@H](O)CO)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
MGAM O43451 4/20 0.38
GAA P10253 4/20 0.38
SI P14410 4/20 0.38
MGAM2 Q2M2H8 4/20 0.38
MAPK14 Q16539 2/20 0.38
MEN1 O00255 3/20 0.36
MAPT P10636 3/20 0.36
KMT2A Q03164 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
MAPK1 P28482 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
SLC6A9 P48067 1/20 0.36
MCL1 Q07820 2/20 0.36
LMNA P02545 1/20 0.36
EPHX2 P34913 1/20 0.36
ACSS2 Q9NR19 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL362902 0.90 GPBAR1 (0.45) BRD4ALDH1A1KDM4EHPGDMAPK14
SCHEMBL364728 0.85 BRD4 (0.42) BRD4ALDH1A1MGAMGAASI
SCHEMBL370940 0.84 BRD4 (0.41) BRD4MGAMGAASIMGAM2
SCHEMBL363956 0.84 BRD4 (0.41) BRD4MGAMGAASIMGAM2
SCHEMBL363934 0.83 GPBAR1 (0.47) BRD4MGAMGAASIMGAM2
SCHEMBL14896301 0.83 BRD4 (0.48) BRD4HPGDMGAMGAASI
SCHEMBL364654 0.83 NPC1 (0.43) BRD4KDM4EMGAMGAASI
SCHEMBL362661 0.81 BRD4 (0.38) BRD4MGAMGAASIMGAM2
SCHEMBL1390288 0.81 BRD4 (0.38) BRD4ALDH1A1KDM4EHPGDMAPK14
SCHEMBL1390287 0.81 BRD4 (0.38) BRD4ALDH1A1KDM4EHPGDMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed