SCHEMBL3644875

SCHEMBL3644875

C[C@@H](CN)N(C)C(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
ALDH1A1 P00352 1/20 0.55
BCAT2 O15382 1/20 0.47
TACR1 P25103 2/20 0.45
SCN1A P35498 3/20 0.45
SCN2A Q99250 3/20 0.45
SCN3A Q9NY46 3/20 0.45
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
KCNH2 Q12809 1/20 0.44
GAA P10253 1/20 0.41
LTB4R2 Q9NPC1 2/20 0.40
CHRNB2 P17787 2/20 0.40
CHRNB4 P30926 2/20 0.40
CHRNA3 P32297 2/20 0.40
CHRNA4 P43681 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3645502 1.00 MEN1 (0.59) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL3647583 1.00 MEN1 (0.59) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL19435298 0.88 MEN1 (0.63) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL17559748 0.88 MEN1 (0.63) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL3640680 0.86 MEN1 (0.56) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL3644829 0.86 MEN1 (0.56) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL3646087 0.86 MEN1 (0.56) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL3644574 0.83 MEN1 (0.54) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL3648367 0.83 MEN1 (0.54) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2
SCHEMBL3649519 0.83 MEN1 (0.54) MEN1KMT2ASMN1; SMN2ALDH1A1BCAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188282-A2 1,2-DIAMIDO-ETHYLENE DERIVATIVES AS OREXIN ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2010-05-26 EP disclosed
WO-2009022311-A2 1,2-DIAMIDO-ETHYLENE DERIVATIVES AS OREXIN ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2009-02-19 WO disclosed