SCHEMBL3649846

SCHEMBL3649846

Cc1ccccc1C1CCN(S(=O)(=O)c2cccnc2)CC1C(=O)N1CCN(c2cc(Cl)ccc2C)CC1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.71
USP2 O75604 3/20 0.71
NPSR1 Q6W5P4 1/20 0.71
SMN1; SMN2 Q16637 6/20 0.53
MAPT P10636 2/20 0.53
POLB P06746 2/20 0.50
ALDH1A1 P00352 2/20 0.49
LMNA P02545 4/20 0.49
TSHR P16473 2/20 0.49
NAMPT P43490 1/20 0.47
THRB P10828 1/20 0.46
KDM4E B2RXH2 1/20 0.45
HSD17B10 Q99714 1/20 0.45
AR P10275 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4219683 1.00 HTT (0.71) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3651413 1.00 HTT (0.71) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3696317 0.91 HTT (0.72) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3692588 0.91 HTT (0.72) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL13269945 0.90 USP2 (0.56) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3653569 0.90 USP2 (0.56) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3650375 0.90 USP2 (0.56) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3650956 0.90 USP2 (0.56) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3692287 0.89 HTT (0.66) HTTUSP2NPSR1SMN1; SMN2MAPT
SCHEMBL3689554 0.89 HTT (0.66) HTTUSP2NPSR1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2188266-A2 NOVEL PIPERAZINE AMIDE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-05-26 EP disclosed
WO-2009021868-A2 NOVEL PIPERAZINE AMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-02-19 WO disclosed