SCHEMBL3652018

SCHEMBL3652018

O=CC(c1cccnc1)c1ccc(Cl)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.46
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 1/20 0.41
CYP3A4 P08684 6/20 0.41
CYP3A5 P20815 6/20 0.41
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
IDO1 P14902 2/20 0.39
SLC6A2 P23975 1/20 0.39
TDO2 P48775 1/20 0.38
KCNA5 P22460 2/20 0.38
KCND3 Q9UK17 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3658241 0.84 KCNA5 (0.45) CYP19A1ALDH1A1LMNASLC6A4SLC6A3
SCHEMBL3658338 0.82 MEN1 (0.46) CYP19A1LMNASLC6A4CYP3A4KMT2A
SCHEMBL11458875 0.82 IDO1 (0.51) LMNAKMT2AMEN1MAPTIDO1
SCHEMBL6501170 0.81 CYP19A1 (0.46) CYP19A1ALDH1A1KDM4EPKMSLC6A4
SCHEMBL6503338 0.80 CYP19A1 (0.62) CYP19A1SLC6A4SLC6A3CYP3A4CYP3A5
SCHEMBL10968603 0.79 CYP19A1 (0.51) CYP19A1ALDH1A1LMNAKDM4EPKM
SCHEMBL2474024 0.78 KCNA5 (0.47) CYP19A1ALDH1A1LMNASLC6A4SLC6A3
SCHEMBL4686827 0.78 TP53 (0.44) CYP19A1LMNAKMT2AMEN1IDO1
SCHEMBL10967991 0.78 SMN1; SMN2 (0.53) CYP19A1ALDH1A1LMNAKDM4EPKM
Hydrochloric Acid SCHEMBL11192967 0.78 CYP19A1 (0.50) CYP19A1ALDH1A1LMNAKDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205562-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. Hoffmann-Roche AG (CH) 2010-07-14 EP disclosed
WO-2009040288-A1 1,1,1-TRIFLUORO-2-HYDROXY-3-PHENYLPROPANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-04-02 WO disclosed