SCHEMBL365209

SCHEMBL365209

CS(=O)(=O)NC(=O)c1cc(F)c(Oc2nncc3ccccc23)cc1F

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 17/20 0.53
HTT P42858 1/20 0.45
SCN5A Q14524 2/20 0.45
ABCB11 O95342 1/20 0.44
CYP2C9 P11712 1/20 0.44
SCN1A P35498 1/20 0.44
SCN4A P35499 1/20 0.44
SCN2A Q99250 1/20 0.44
SCN3A Q9NY46 1/20 0.44
SCN8A Q9UQD0 1/20 0.44
SCN10A Q9Y5Y9 1/20 0.44
POLB P06746 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL363677 0.84 SCN9A (0.53) SCN9ASCN5AABCB11CYP2C9SCN1A
SCHEMBL1690177 0.78 SCN9A (0.68) SCN9ASCN5AABCB11CYP2C9SCN1A
SCHEMBL16175029 0.78 SCN9A (0.56) SCN9ASCN5A
SCHEMBL365248 0.78 SCN9A (0.53) SCN9A
SCHEMBL679301 0.77 SCN9A (0.63) SCN9ASCN5AABCB11CYP2C9SCN1A
SCHEMBL365882 0.77 SCN9A (0.53) SCN9ASCN5AABCB11CYP2C9SCN1A
SCHEMBL1690176 0.76 SCN9A (0.53) SCN9ASCN5AABCB11CYP2C9SCN1A
SCHEMBL1690173 0.76 SCN9A (0.58) SCN9ASCN5A
SCHEMBL1690225 0.76 SCN9A (0.60) SCN9ASCN5ASCN1A
SCHEMBL680139 0.75 SCN9A (0.61) SCN9ASCN5AABCB11CYP2C9SCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593432-B1 N-SULFONYLBENZAMIDE DERIVATIVES USEFUL AS VOLTAGE GATED SODIUM CHANNEL INHIBITORS PFIZER LTD (GB) 2014-10-22 EP disclosed
US-8592629-B2 Sulfonamide derivatives as Nav 1.7 inhibitors PFIZER LIMITED (GB) 2013-11-26 US disclosed
EP-2593432-A1 N-SULFONYLBENZAMIDE DERIVATIVES USEFUL AS VOLTAGE GATED SODIUM CHANNEL INHIBITORS Pfizer Limited (GB) 2013-05-22 EP disclosed
WO-2012007861-A1 N-SULFONYLBENZAMIDE DERIVATIVES USEFUL AS VOLTAGE GATED SODIUM CHANNEL INHIBITORS PFIZER LIMITED (GB) 2012-01-19 WO disclosed
US-20120010183-A1 Chemical Compounds PFIZER LIMITED (GB) 2012-01-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010183-A1 Chemical Compounds SCN1A, SCN1B, SCN7A SCN9A 25/4885HTT 655/4885SCN5A 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.