SCHEMBL3655587

SCHEMBL3655587

O=C(OCc1ccccc1)C1CN(C(=O)O)CCN1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
BACE1 P56817 1/20 0.44
CYP2C19 P33261 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
GLA P06280 1/20 0.41
HTR2C P28335 1/20 0.41
FABP7 O15540 1/20 0.41
FABP5 Q01469 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
FKBP1A P62942 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10281640 0.90 TSHR (0.48) TSHRSMN1; SMN2NPC1RAB9ABACE1
SCHEMBL2680993 0.87 CHRM5 (0.43) TSHRSMN1; SMN2NPC1RAB9AMEN1
SCHEMBL17153132 0.86 JAK2 (0.47) TSHRMEN1KMT2A
SCHEMBL20418703 0.83 TSHR (0.59) TSHRSMN1; SMN2NPC1RAB9ABACE1
SCHEMBL629930 0.83 TSHR (0.59) TSHRSMN1; SMN2NPC1RAB9ABACE1
SCHEMBL15251729 0.83 TSHR (0.59) TSHRSMN1; SMN2NPC1RAB9ABACE1
SCHEMBL12324603 0.83 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL14646669 0.83 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
SCHEMBL2680992 0.83 SMN1; SMN2 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19MEN1
Hydrochloric Acid SCHEMBL29121517 0.82 SMN1; SMN2 (0.51) TSHRSMN1; SMN2NPC1RAB9ACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1976904-A Pyridazin-3 (2H) -one derivatives and their use as PDE4 inhibitors ALMIRALL LAB (ES) 2007-06-06 CN claimed
EP-2217600-A2 FUNGICIDAL BICYCLIC PYRAZOLES E. I. du Pont de Nemours and Company (US) 2010-08-18 EP disclosed
WO-2009076440-A2 FUNGICIDAL BICYCLIC PYRAZOLES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2009-06-18 WO disclosed
CN-1976904-A Pyridazin-3 (2H) -one derivatives and their use as PDE4 inhibitors ALMIRALL LAB (ES) 2007-06-06 CN disclosed