SCHEMBL3657993

SCHEMBL3657993

CC(N)CCc1cccs1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.55
ADRA2A P08913 3/20 0.46
ADRA2B P18089 3/20 0.46
ADRA2C P18825 3/20 0.46
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43
RAB9A P51151 1/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
TSHR P16473 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 2/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.39
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
CTSC P53634 2/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10667983 0.89 TAAR1 (0.57) TAAR1ADRA2AADRA2BADRA2CRAB9A
Hydrochloric Acid SCHEMBL7533264 0.87 TAAR1 (0.55) TAAR1ADRA2AADRA2BADRA2CRAB9A
SCHEMBL4729505 0.83 TAAR1 (0.54) TAAR1ADRA2AADRA2BADRA2CRAB9A
SCHEMBL5168937 0.82 TAAR1 (0.48) TAAR1ADRA2AADRA2BADRA2CRAB9A
SCHEMBL4210706 0.82 TAAR1 (0.48) TAAR1ADRA2AADRA2BADRA2CRAB9A
Ammonia Solution, Strong SCHEMBL28852825 0.82 TAAR1 (0.52) TAAR1ADRA2AADRA2BADRA2CRAB9A
SCHEMBL7534232 0.81 TAAR1 (0.52) TAAR1ADRA2AADRA2BADRA2CRAB9A
SCHEMBL7534237 0.81 TAAR1 (0.52) TAAR1ADRA2AADRA2BADRA2CRAB9A
SCHEMBL23094084 0.80 TAAR1 (0.50) TAAR1ADRA2AADRA2BADRA2CRAB9A
SCHEMBL10728212 0.80 KMT2A (0.50) TAAR1ADRA2AADRA2BADRA2CRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110669058-A Tricyclic quinolone carboxylic acid and preparation method thereof 江西农业大学 2020-01-10 CN claimed
WO-2020035070-A1 3-ARYLOXY-3-ARYL-PROPYLAMINE COMPOUND AND USES THEREOF 漳州片仔癀药业股份有限公司 2020-02-20 WO disclosed
CN-110669058-A Tricyclic quinolone carboxylic acid and preparation method thereof 江西农业大学 2020-01-10 CN disclosed
EP-2205589-A2 C-MET PROTEIN KINASE INHIBITORS Vertex Pharmaceuticals Incorporated (US) 2010-07-14 EP disclosed
WO-2009045992-A2 C-MET PROTEIN KINASE INHIBITORS VERTEX PHARMACEUTICALS INCORPORATED (US) 2009-04-09 WO disclosed
WO-2007023281-A2 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2007-03-01 WO disclosed
EP-1622867-A1 N-(2-PHENYLETHYL)SULFAMIDE DERIVATIVES AS INTEGRIN ALPHA4 ANTAGONISTS Almirall Prodesfarma, S.A. (ES) 2006-02-08 EP disclosed
WO-2004099126-A1 N-(2-PHENYLETHYL)SULFAMIDE DERIVATIVES AS INTEGRIN α4 ANTAGONISTS ALMIRALL PRODESFARMA SA (ES) 2004-11-18 WO disclosed
US-4242474-A A POLYHYDROXY ACRYLIC ESTER REACTED WITH AN ISOCYANATE TERMINATED POLYOXYALKYLENE GLYCOL; BIOPOLYMERS TERUMO CORPORATION (JP) 1980-12-30 US disclosed