SCHEMBL3658274

SCHEMBL3658274

CC(C(=O)O)c1ccc(NC(=O)C(C2CCCCC2)C2(c3ccc(Cl)cc3)Nc3cc(F)c(F)cc3N2)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 10/20 0.41
CYP2C9 P11712 5/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
KCNH2 Q12809 2/20 0.40
APP P05067 3/20 0.39
LMNA P02545 2/20 0.38
MAPT P10636 1/20 0.38
FAAH O00519 3/20 0.38
TP53 P04637 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3659255 0.89 NR1H4 (0.39) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3658772 0.86 NR1H4 (0.44) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3656457 0.86 NR1H4 (0.55) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3654621 0.84 NR1H4 (0.41) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3653472 0.83 NR1H4 (0.45) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3652400 0.82 NR1H4 (0.40) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3649203 0.82 NR1H4 (0.42) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3651277 0.82 NR1H4 (0.57) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3659323 0.82 NR1H4 (0.57) NR1H4CYP2C9CYP3A4CYP2D6KCNH2
SCHEMBL3660110 0.82 NR1H4 (0.43) NR1H4CYP2C9CYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225221-A2 CARBOXYL- OR HYDROXYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2010-09-08 EP claimed
WO-2009080555-A2 CARBOXYL- OR HYDROXYL- SUBSTITUTED BENZIMIDAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-07-02 WO claimed