SCHEMBL3658730

SCHEMBL3658730

CCc1c(Cc2ccc(F)c(C(=O)N3CCN(C4CCCCC4)C(=O)C3)c2)n[nH]c(=O)c1C(F)(F)F

nearest known ligand 0.56

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.56
PARP2 Q9UGN5 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3081532 0.97 PARP1 (0.53) PARP1PARP2
SCHEMBL15988465 0.92 PARP1 (0.57) PARP1PARP2
SCHEMBL15988423 0.90 PARP1 (0.58) PARP1PARP2
SCHEMBL15988435 0.90 PARP1 (0.58) PARP1PARP2
Trifluoroacetic Acid SCHEMBL3063430 0.89 PARP1 (0.54) PARP1PARP2
Trifluoroacetic Acid SCHEMBL3082902 0.89 PARP1 (0.54) PARP1PARP2
Trifluoroacetic Acid SCHEMBL3083043 0.89 PARP1 (0.54) PARP1PARP2
SCHEMBL15988392 0.86 PARP1 (0.67) PARP1
SCHEMBL12342209 0.86 PARP1 (0.67) PARP1
SCHEMBL30418013 0.85 PARP1 (0.68) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2220073-B1 PYRIDAZINONE DERIVATIVES AS PARP INHIBITORS MSD ITALIA SRL (IT) 2014-09-03 EP claimed
EP-2220073-A1 PYRIDAZINONE DERIVATIVES AS PARP INHIBITORS Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. (IT) 2010-08-25 EP disclosed
WO-2009063244-A1 PYRIDAZINONE DERIVATIVES AS PARP INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2009-05-22 WO disclosed