SCHEMBL3658734

SCHEMBL3658734

O=C(Nc1ccc(-c2nc(N3C4CCC3COC4)c3cnn(C4CCN(C(=O)O)CC4)c3n2)cc1)Nc1ccc(N2CCNCC2)cc1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 20/20 0.67
MTOR P42345 20/20 0.67
PIK3CG P48736 3/20 0.55
ATR Q13535 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL55731 0.92 PIK3CA (0.80) PIK3CAMTORPIK3CGATR
SCHEMBL53026 0.85 PIK3CA (0.83) PIK3CAMTORPIK3CGATR
SCHEMBL55405 0.83 PIK3CA (0.77) PIK3CAMTOR
SCHEMBL3654553 0.83 PIK3CA (0.65) PIK3CAMTORPIK3CG
SCHEMBL55818 0.82 PIK3CA (0.87) PIK3CAMTORPIK3CGATR
Hydrochloric Acid SCHEMBL56134 0.82 PIK3CA (0.76) PIK3CAMTOR
SCHEMBL4563300 0.81 PIK3CA (0.78) PIK3CAMTORPIK3CGATR
SCHEMBL56098 0.80 PIK3CA (0.86) PIK3CAMTORPIK3CGATR
SCHEMBL55501 0.80 PIK3CA (1.00) PIK3CAMTORPIK3CGATR
SCHEMBL3983804 0.80 PIK3CA (0.75) PIK3CAMTORPIK3CGATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212333-A1 THIENOPYRIMIDINE AND PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS Wyeth LLC (US) 2010-08-04 EP disclosed
WO-2009052145-A1 THIENOPYRIMIDINE AND PYRAZOLOPYRIMIDINE COMPOUNDS AND THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS WYETH (US) 2009-04-23 WO disclosed