SCHEMBL3663268

SCHEMBL3663268

Cc1nn(-c2cc(F)c(C(N)=O)c(N[C@H]3CCCCC3N)c2)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 18/20 0.55
HSP90AA1 P07900 16/20 0.55
HSP90B1 P14625 4/20 0.51
TRAP1 Q12931 3/20 0.51
OPRM1 P35372 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5004864 1.00 HSP90AB1 (0.55) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL5004866 1.00 HSP90AB1 (0.55) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL8132799 0.92 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL3632672 0.92 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL8132369 0.90 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL8139260 0.90 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL5005349 0.90 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL3626162 0.90 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1OPRM1
SCHEMBL3632747 0.90 HSP90AB1 (0.65) HSP90AB1HSP90AA1HSP90B1TRAP1
SCHEMBL3624481 0.90 HSP90AB1 (0.57) HSP90AB1HSP90AA1HSP90B1TRAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2146967-A2 TETRAHYDROINDOLE AND TETRAHYDROINDAZOLE DERIVATIVES Serenex, Inc. (US) 2010-01-27 EP disclosed
WO-2008130879-A2 TETRAHYDROINDOLE AND TETRAHYDROINDAZOLE DERIVATIVES SERENEX, INC. (US) 2008-10-30 WO disclosed