SCHEMBL3663796

SCHEMBL3663796

FCOc1cccc(CCBr)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.45
CYP4A11 Q02928 1/20 0.45
TDP1 Q9NUW8 1/20 0.43
KCNH2 Q12809 1/20 0.42
MAOB P27338 3/20 0.41
TAAR1 Q96RJ0 1/20 0.41
MGLL Q99685 1/20 0.39
CHRM2 P08172 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
BCHE P06276 4/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2368219 0.85 MAOB (0.43) CYP4F2CYP4A11KCNH2MAOBBCHE
SCHEMBL28822312 0.81 CETP (0.43) CYP4F2CYP4A11TDP1KCNH2MAOB
SCHEMBL13715411 0.80 BCHE (0.42) CYP4F2CYP4A11KCNH2MAOBTAAR1
SCHEMBL27733468 0.80 CYP4F2 (0.70) CYP4F2CYP4A11MAOBMGLLBCHE
SCHEMBL27721818 0.77 BCHE (0.49) CYP4F2CYP4A11TDP1CHRM2CHRM1
SCHEMBL9621361 0.77 CYP2D6 (0.53) KCNH2PPARGPPARA
SCHEMBL27825974 0.77 KDM4E (0.48) CYP4F2CYP4A11MAOBTAAR1CHRM2
SCHEMBL4737237 0.77 TP53 (0.45) MAOB
SCHEMBL9442243 0.77 MAOB (0.44) TDP1KCNH2MAOB
SCHEMBL177862 0.77 TAAR1 (0.67) TAAR1CHRM2CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217598-A1 NEW TETRACYCLIC COMPOUNDS Medivation Technologies, Inc. (US) 2010-08-18 EP disclosed
WO-2009055828-A1 NEW TETRACYCLIC COMPOUNDS MEDIVATION TECHNOLOGIES, INC. (US) 2009-04-30 WO disclosed