SCHEMBL3665008

SCHEMBL3665008

COCC(=O)N1CCC(Oc2cc3c(Nc4ccc(F)c(Cl)c4)ncnc3cc2OC)CC1.COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OC1CCCNC1

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 5/20 0.65
EGFR P00533 17/20 0.65
KDR P35968 2/20 0.56
EPHB4 P54760 2/20 0.56
EPHA2 P29317 1/20 0.56
AURKA O14965 1/20 0.54
INSR P06213 1/20 0.54
FBP1 P09467 1/20 0.54
PDGFRB P09619 1/20 0.54
FLT4 P35916 1/20 0.54
CLK1 P49759 1/20 0.54
TEK Q02763 1/20 0.54
AURKB Q96GD4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL118271 0.93 EGFR (0.75) ERBB2EGFRKDREPHB4EPHA2
SCHEMBL29623483 0.93 EGFR (0.75) ERBB2EGFRKDREPHB4EPHA2
SCHEMBL12743401 0.88 EGFR (0.73) ERBB2EGFRKDREPHB4EPHA2
SCHEMBL29623405 0.88 EGFR (0.72) ERBB2EGFRKDREPHB4EPHA2
SCHEMBL186250 0.88 EGFR (0.72) ERBB2EGFRKDREPHB4EPHA2
SCHEMBL1943054 0.88 EGFR (0.77) ERBB2EGFRKDREPHB4AURKA
Hydrochloric Acid SCHEMBL1446449 0.87 EGFR (0.71) ERBB2EGFRKDREPHB4EPHA2
SCHEMBL4421677 0.87 EGFR (0.69) ERBB2EGFRKDREPHB4EPHA2
SCHEMBL1446188 0.87 ERBB2 (0.66) ERBB2EGFRFBP1
SCHEMBL2762294 0.87 EGFR (0.67) ERBB2EGFRKDREPHB4EPHA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2146764-A2 DISPENSING DEVICE Boehringer Ingelheim International GmbH (DE) 2010-01-27 EP disclosed
WO-2008138628-A2 DISPENSING DEVICE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-11-20 WO disclosed