SCHEMBL3670577

SCHEMBL3670577

C1=COCCNCCNCCN1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
CYP2C9 P11712 1/20 0.39
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HIF1A Q16665 1/20 0.30
MAPT P10636 1/20 0.30
PDE4A P27815 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morpholine SCHEMBL10437036 0.86 MEN1 (0.48) KDM4EGAACYP2C9MEN1KMT2A
SCHEMBL441202 0.84
SCHEMBL19956080 0.79 MEN1 (0.52) KDM4EGAACYP2C9MEN1KMT2A
SCHEMBL30146940 0.78 MEN1 (0.44) KDM4EGAACYP2C9MEN1KMT2A
SCHEMBL1830024 0.74
SCHEMBL17319684 0.72
Morpholine SCHEMBL1808505 0.71 MEN1 (0.48) KDM4EGAACYP2C9MEN1KMT2A
SCHEMBL1782105 0.71 HIF1A (0.50) KDM4EGAACYP2C9HIF1AMAPT
SCHEMBL1781839 0.71 HIF1A (0.50) KDM4EGAACYP2C9HIF1AMAPT
SCHEMBL1780932 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111808161-A Method for radiolabeling biological compounds 北京大学 2020-10-23 CN claimed
CN-104710504-A Methods for generating radioimmunoconjugates ACTINIUM PHARMACEUTICALS INC 2015-06-17 CN claimed
CN-101674807-B Compositions for reducing, ameliorating, treating, or preventing dry eye, and methods of making and using same BAUSCH & LOMB 2013-03-20 CN claimed
CN-114728074-A Radiolabeling of anti-CD 45 immunoglobulins and methods of use thereof 锕医药有限责任公司 2022-07-08 CN disclosed
CN-113195006-A Combination therapy of radioimmunotherapy and immunodetection point therapy for the treatment of cancer 锕医药有限责任公司 2021-07-30 CN disclosed
CN-111808161-A Method for radiolabeling biological compounds 北京大学 2020-10-23 CN disclosed
CN-111050796-A Treatment of hematologic malignancies 锕医药股份有限公司 2020-04-21 CN disclosed
CN-105377287-A Kit for tumor imaging UNIV JEFFERSON 2016-03-02 CN disclosed
CN-104710504-A Methods for generating radioimmunoconjugates ACTINIUM PHARMACEUTICALS INC 2015-06-17 CN disclosed
CN-102596258-B Method for preparing a radioactive immunoconjugate ACTINIUM PHARMACEUTICALS INC 2015-01-28 CN disclosed
CN-101674807-B Compositions for reducing, ameliorating, treating, or preventing dry eye, and methods of making and using same BAUSCH & LOMB 2013-03-20 CN disclosed
WO-2010016858-A2 MOLECULAR IMAGING PROBES CARESTREAM HEALTH, INC. (US) 2010-02-11 WO disclosed
EP-2148701-A2 IMAGING CONTRAST AGENTS USING NANOPARTICLES Carestream Health, Inc. (US) 2010-02-03 EP disclosed
WO-2008140475-A2 IMAGING CONTRAST AGENTS USING NANOPARTICLES CARESTREAM HEALTH, INC. (US) 2008-11-20 WO disclosed
US-20020072667-A1 MAGNETIC RESONANCE IMAGING KUCHARCZYK JOHN (US) 2002-06-13 US disclosed