SCHEMBL3671935

SCHEMBL3671935

Cc1cc2c(-c3ccc(S(=O)(=O)NCC(NC(=O)O)C(C)(C)C)s3)ccnc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 1/20 0.39
PTGDR2 Q9Y5Y4 3/20 0.37
PIK3C3 Q8NEB9 1/20 0.36
CAPN1 P07384 7/20 0.35
MMP13 P45452 3/20 0.34
MMP1 P03956 2/20 0.34
MCL1 Q07820 1/20 0.33
PFKFB3 Q16875 2/20 0.33
ENPP3 O14638 1/20 0.32
ENPP1 P22413 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2984751 0.82 MAP3K5 (0.43) MAP3K5PTGDR2PIK3C3CAPN1MCL1
SCHEMBL13241039 0.81 P2RY14 (0.43) MAP3K5PTGDR2CAPN1MCL1KDM4E
SCHEMBL4317149 0.79 IKBKB (0.40) PTGDR2PIK3C3MMP13
SCHEMBL13241037 0.78 PTGDR2 (0.40) MAP3K5PTGDR2PIK3C3
SCHEMBL13981531 0.77 CA12 (0.48) MAP3K5PTGDR2PIK3C3
Trifluoroacetic Acid SCHEMBL3633505 0.76 MAP3K5 (0.59) MAP3K5
SCHEMBL2987892 0.74 IKBKB (0.38) MAP3K5PTGDR2PIK3C3MMP13MMP1
SCHEMBL2987895 0.73 IKBKB (0.45) MAP3K5PTGDR2PIK3C3
SCHEMBL2980723 0.73 MAP3K5 (0.52) MAP3K5PTGDR2CAPN1MCL1
SCHEMBL13241054 0.69 PTGDR2 (0.36) MAP3K5PTGDR2PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2162455-A2 PYRROLOPYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS MEDICAMENTS Glaxo Group Limited (GB) 2010-03-17 EP disclosed
WO-2008145688-A2 PYRROLOPYRIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR USE AS MEDICAMENTS GLAXO GROUP LIMITED (GB) 2008-12-04 WO disclosed