SCHEMBL3672959

SCHEMBL3672959

CC1COCCN1c1nc(Cl)nc2c1CCN(C(=O)O)C2

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 7/20 0.53
MTOR P42345 13/20 0.47
KCNH2 Q12809 1/20 0.47
PIK3CA P42336 1/20 0.47
RPTOR Q8N122 5/20 0.45
MLST8 Q9BVC4 5/20 0.45
CYP3A4 P08684 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1831760 0.92 ATR (0.47) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL441654 0.91 MTOR (0.47) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL2097798 0.88 ATR (0.52) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL1829520 0.88 ATR (0.52) ATRMTORKCNH2PIK3CARPTOR
SCHEMBL24955630 0.86 MTOR (0.55) ATRMTORPIK3CA
SCHEMBL442685 0.86 MTOR (0.55) ATRMTORPIK3CA
SCHEMBL31107005 0.86 MTOR (0.55) ATRMTORPIK3CA
SCHEMBL412512 0.86 MTOR (0.55) ATRMTORPIK3CA
SCHEMBL443375 0.84 MTOR (0.51) ATRMTORKCNH2PIK3CACYP3A4
SCHEMBL414101 0.84 MTOR (0.51) ATRMTORKCNH2PIK3CACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010103094-A1 PYRIMIDINE DERIVATIVES AS mTOR INHIBITORS CELLZOME LIMITED (GB) 2010-09-16 WO disclosed