Theracys

Theracys

SCHEMBL367470

CN1C2CC[C@H]1CC(OC(=O)c1ccccc1)C2C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.80
SLC6A2 P23975 2/20 0.80
SLC6A4 P31645 2/20 0.80
SLC6A3 Q01959 2/20 0.80
MAPT P10636 1/20 0.80
MAOA P21397 1/20 0.80
SCN1A P35498 1/20 0.80
SCN2A Q99250 1/20 0.80
SIGMAR1 Q99720 1/20 0.80
SCN3A Q9NY46 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Theracys SCHEMBL18648964 1.00 KCNH2 (0.80) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL328884 1.00 KCNH2 (0.80) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL116803 1.00 KCNH2 (0.80) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL13196454 1.00 KCNH2 (0.80) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL16922152 1.00 KCNH2 (0.80) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL328885 1.00 KCNH2 (0.80) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL11415956 0.99 KCNH2 (0.78) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL6716416 0.99 SLC6A2 (0.80) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Theracys SCHEMBL8958743 0.94 KCNH2 (0.72) KCNH2SLC6A2SLC6A4SLC6A3MAPT
Cocaine SCHEMBL8050369 0.93 KCNH2 (0.93) KCNH2SLC6A2SLC6A4SLC6A3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012009263-A1 COCAINE ANALOGS AND METHODS OF PREPARATION AND USES THEREOF TEMPLE UNIVERSITY-OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2012-01-19 WO disclosed