SCHEMBL3676766

SCHEMBL3676766

CCc1cccc(NC(=O)c2ccc(N3CCCC3)c(C(F)(F)F)c2)c1.COc1cccc(NC(=O)c2ccc(N3CCOCC3)c(C(F)(F)F)c2)c1

nearest known ligand 0.77

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.69
TP53 P04637 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
MAPT P10636 1/20 0.60
THRB P10828 1/20 0.60
RAF1 P04049 1/20 0.58
BRAF P15056 1/20 0.58
NPC1 O15118 1/20 0.54
LMNA P02545 1/20 0.54
RAB9A P51151 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4248596 0.91 SMN1; SMN2 (0.71) TAAR1TP53SMN1; SMN2MAPTTHRB
SCHEMBL3638666 0.88 TAAR1 (0.74) TAAR1TP53SMN1; SMN2MAPTTHRB
SCHEMBL4247984 0.88 TAAR1 (0.80) TAAR1TP53SMN1; SMN2MAPTTHRB
SCHEMBL3642495 0.87 TAAR1 (0.79) TAAR1
SCHEMBL3645668 0.87 TAAR1 (0.79) TAAR1
SCHEMBL3645506 0.86 TAAR1 (0.77) TAAR1TP53SMN1; SMN2MAPTTHRB
SCHEMBL29690457 0.82 TAAR1 (1.00) TAAR1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL3647615 0.82 TAAR1 (1.00) TAAR1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL4254287 0.81 TAAR1 (0.68) TAAR1RAF1BRAF
SCHEMBL4254100 0.81 TAAR1 (0.77) TAAR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2182935-A1 THE USE OF BENZAMIDE DERIVATIVES FOR THE TREATMENT OF CNS DISORDERS F. Hoffmann-Roche AG (CH) 2010-05-12 EP disclosed
WO-2009016088-A1 THE USE OF BENZAMIDE DERIVATIVES FOR THE TREATMENT OF CNS DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 WO disclosed