SCHEMBL3679645

SCHEMBL3679645

CC(C)(C)OC(=O)CC(CI)NC(=O)OC(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.54
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CTSK P43235 11/20 0.42
ATM Q13315 1/20 0.40
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
CTSS P25774 5/20 0.38
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC8 Q9BY41 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16970605 1.00 CYP2D6 (0.54) CYP2D6CA1CA2CA7CTSK
SCHEMBL3679648 1.00 CYP2D6 (0.54) CYP2D6CA1CA2CA7CTSK
SCHEMBL22231132 0.92 CYP2D6 (0.45) CYP2D6CA1CA2CA7CTSK
SCHEMBL13230319 0.92 CYP2D6 (0.45) CYP2D6CA1CA2CA7CTSK
SCHEMBL16970731 0.92 CYP2D6 (0.45) CYP2D6CA1CA2CA7CTSK
SCHEMBL28520968 0.87 CYP2D6 (0.51) CYP2D6CA1CA2CA7CTSK
SCHEMBL28520969 0.87 CYP2D6 (0.51) CYP2D6CA1CA2CA7CTSK
SCHEMBL16974993 0.86 CA1 (0.44) CYP2D6CA1CA2CA7CTSK
SCHEMBL16974944 0.86 CA1 (0.44) CYP2D6CA1CA2CA7CTSK
SCHEMBL18445855 0.86 CA1 (0.44) CYP2D6CA1CA2CA7CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026026-B Beta-substituted beta-amino acids and analogs as chemotherapeutic agents and uses thereof 夸德里加生物科学公司 2021-02-09 CN disclosed
US-8410150-B2 Inhibitors of carnitine palmitoyltransferase and treating cancer UNIVERSITY HEALTH NETWORK (CA) 2013-04-02 US disclosed
US-20100105900-A1 INHIBITORS OF CARNITINE PALMITOYLTRANSFERASE AND TREATING CANCER UNIVERSITY HEALTH NETWORK 2010-04-29 US disclosed
WO-2008109991-A1 INHIBITORS OF CARNITINE PALMITOYLTRANSFERASE AND TREATING CANCER UNIVERSITY HEALTH NETWORK (CA) 2008-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100105900-A1 INHIBITORS OF CARNITINE PALMITOYLTRANSFERASE AND TREATING CANCER CPT1A, CPT1B, CPT2 CYP2D6 1791/4885CA1 1983/4885CA2 1295/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.