SCHEMBL3686706

SCHEMBL3686706

COC(=O)C(OP(=O)(O)[C@@H](NS(=O)(=O)Cc1ccccc1)C(C)C)c1cccc(N(C(=O)OC(C)(C)C)C(N)=NC(=O)OC(C)(C)C)c1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 1/20 0.32
ITGB1 P05556 1/20 0.30
ITGA4 P13612 1/20 0.30
BACE1 P56817 1/20 0.30
STS P08842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696034 0.94 ITGB1 (0.32) CNR1ITGB1ITGA4BACE1STS
SCHEMBL2349106 0.87 BACE1 (0.39) BACE1
SCHEMBL3690224 0.87 BACE1 (0.39) BACE1
SCHEMBL3687462 0.83 ITGB1 (0.30) ITGB1ITGA4
SCHEMBL3688466 0.83 ITGB1 (0.30) ITGB1ITGA4
SCHEMBL2352504 0.82 BACE1 (0.40) BACE1
SCHEMBL3688178 0.81 HTT (0.35)
SCHEMBL2349221 0.74 BACE1 (0.34) BACE1STS
SCHEMBL2349103 0.73 BACE1 (0.40) BACE1
SCHEMBL3688119 0.73 ITGB1 (0.31) ITGB1ITGA4BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2204373-A1 Phosphonic acid as Plasma Carboxypeptidase B Inhibitors Bayer Schering Pharma Aktiengesellschaft (DE) 2010-07-07 EP disclosed