SCHEMBL3686777

SCHEMBL3686777

Cc1ccccc1-c1ccc(N2CCN(CCO)CC2)c(C=CC(=O)c2ccccc2CN(C)C)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.37
CD274 Q9NZQ7 2/20 0.37
BACE1 P56817 4/20 0.37
NMT2 O60551 1/20 0.37
NMT1 P30419 1/20 0.37
HTR7 P34969 3/20 0.36
DRD2 P14416 3/20 0.36
HTR1A P08908 1/20 0.36
HTR6 P50406 1/20 0.36
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HDAC3 O15379 3/20 0.35
HDAC4 P56524 3/20 0.35
HDAC1 Q13547 3/20 0.35
HDAC7 Q8WUI4 3/20 0.35
HDAC2 Q92769 3/20 0.35
HDAC10 Q969S8 3/20 0.35
HDAC11 Q96DB2 3/20 0.35
HDAC8 Q9BY41 3/20 0.35
HDAC6 Q9UBN7 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3681669 0.91 HDAC3 (0.41) NMT2NMT1DRD2HDAC3HDAC4
SCHEMBL3686776 0.90 PDCD1 (0.39) PDCD1CD274BACE1NMT2NMT1
SCHEMBL3688464 0.90 PDCD1 (0.39) PDCD1CD274BACE1NMT2NMT1
SCHEMBL3681137 0.84 SMYD2 (0.36) PDCD1CD274NMT2NMT1L3MBTL1
SCHEMBL3681667 0.81 HDAC3 (0.41) PDCD1CD274NMT2NMT1DRD2
SCHEMBL3693429 0.81 HDAC3 (0.41) PDCD1CD274NMT2NMT1DRD2
SCHEMBL4852464 0.80 BACE1 (0.50) BACE1DRD2HRH1DRD3MEN1
SCHEMBL3691047 0.79 MEN1 (0.37) PDCD1CD274DRD2MAPTNPSR1
SCHEMBL3690513 0.79 HDAC3 (0.35) PDCD1CD274BACE1NMT2NMT1
SCHEMBL4854149 0.79 BACE1 (0.52) BACE1MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US claimed
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed
EP-1506158-A2 DIAMINO-FUNCTIONAL CHALCONES Lica Pharmaceuticals A/S (DK) 2005-02-16 EP disclosed
WO-2003097576-A2 DIAMINO-FUNCTIONAL CHALCONES LICA PHARMACEUTICALS A/S (DK) 2003-11-27 WO disclosed