SCHEMBL3687310

SCHEMBL3687310

COc1ccc(/C=C/C(=O)c2ccc(NCCN(C)C)cc2)c(OC)c1OC

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 3/20 0.67
CYP1A1 P04798 2/20 0.58
CYP1A2 P05177 2/20 0.58
CYP2D6 P10635 2/20 0.58
CYP1B1 Q16678 2/20 0.58
CYP3A4 P08684 1/20 0.51
CHRNA7 P36544 1/20 0.48
LMNA P02545 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
ALOX5 P09917 1/20 0.48
TP53 P04637 1/20 0.48
MAOB P27338 1/20 0.47
CTSL P07711 2/20 0.45
CTSB P07858 2/20 0.45
MAPT P10636 2/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MITF O75030 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3693509 1.00 ABCG2 (0.67) ABCG2CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL3687801 0.84 TNFRSF1A (0.67) ABCG2CYP1A1CYP1B1LMNASMN1; SMN2
SCHEMBL5915769 0.83 ABCG2 (0.72) ABCG2CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL5915479 0.83 ABCG2 (0.72) ABCG2CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL4855944 0.81 ABCG2 (0.69) ABCG2CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL4852275 0.81 ABCG2 (0.69) ABCG2CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL7102316 0.81 ABCG2 (0.82) ABCG2CYP1A1CYP1A2CYP2D6CYP1B1
SCHEMBL3684939 0.81 TNFRSF1A (0.54) ABCG2LMNASMN1; SMN2NPC1RAB9A
SCHEMBL3687313 0.80 TUBB1 (0.58) ABCG2CYP1A1CYP1A2CYP1B1CYP3A4
SCHEMBL3686109 0.80 MAOB (0.53) ABCG2CYP1A1CYP1B1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed