SCHEMBL3690597

SCHEMBL3690597

Cc1ccccc1-c1ccc(N2CCC(N3CCCC3)CC2)c(C(=O)/C=C/c2ccccc2CN(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.36
SMYD2 Q9NRG4 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
HRH3 Q9Y5N1 2/20 0.35
PDCD1 Q15116 2/20 0.35
CD274 Q9NZQ7 2/20 0.35
L3MBTL3 Q96JM7 4/20 0.35
L3MBTL1 Q9Y468 4/20 0.35
MBTD1 Q05BQ5 1/20 0.34
TP53BP1 Q12888 1/20 0.34
NPY2R P49146 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
CALCA P06881 1/20 0.34
KDM2B Q8NHM5 1/20 0.33
SLC2A1 P11166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3681135 1.00 PTPN1 (0.36) PTPN1SMYD2TDP1HRH3PDCD1
SCHEMBL3681137 0.91 SMYD2 (0.36) PTPN1SMYD2TDP1HRH3PDCD1
SCHEMBL3681667 0.87 HDAC3 (0.41) PTPN1PDCD1CD274TSHR
SCHEMBL3693429 0.87 HDAC3 (0.41) PTPN1PDCD1CD274TSHR
SCHEMBL3686776 0.84 PDCD1 (0.39) PTPN1PDCD1CD274L3MBTL1
SCHEMBL3688464 0.84 PDCD1 (0.39) PTPN1PDCD1CD274L3MBTL1
SCHEMBL3681669 0.78 HDAC3 (0.41) PTPN1TSHR
SCHEMBL3690816 0.78 MCHR1 (0.35) PDCD1CD274POLB
SCHEMBL3690510 0.78 MCHR1 (0.35) PDCD1CD274POLB
SCHEMBL4855930 0.76 BACE1 (0.49) TDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642367-B2 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2010-01-05 US disclosed
US-20060235073-A1 Diamino-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2006-10-19 US disclosed