SCHEMBL3698155

SCHEMBL3698155

COc1ccc(S(=O)(=O)c2cc(CN(C)C(=O)OC(C)(C)C)nn2-c2ccccc2Cl)cn1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.41
SLC6A4 P31645 7/20 0.41
SLC16A3 O15427 8/20 0.38
SLC16A1 P53985 7/20 0.38
AVPR2 P30518 1/20 0.36
OXTR P30559 1/20 0.36
AVPR1A P37288 1/20 0.36
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
TSHR P16473 1/20 0.34
TAS2R14 Q9NYV8 1/20 0.34
HTR2A P28223 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3696906 0.91 HTR2C (0.43) HTR2CSLC6A4SLC16A3SLC16A1ALDH1A1
Fumaric Acid SCHEMBL3706208 0.91 HTR2C (0.37) HTR2CSLC6A4SLC16A3SLC16A1AVPR2
SCHEMBL3805207 0.90 HTR2C (0.39) HTR2CSLC6A4SLC16A3SLC16A1AVPR2
SCHEMBL3696612 0.90 HTR2C (0.42) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL4126439 0.89 KMT2A (0.40) SLC16A3SLC16A1AVPR2OXTRAVPR1A
SCHEMBL3691768 0.85 HTR2C (0.42) HTR2CSLC6A4SLC16A3SLC16A1
SCHEMBL3701580 0.85 HTR2C (0.44) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3698156 0.85 KMT2A (0.38) SLC16A3SLC16A1AVPR2OXTRAVPR1A
SCHEMBL3696893 0.83 SLC16A3 (0.46) HTR2CSLC6A4SLC16A3SLC16A1HTR2A
SCHEMBL3698587 0.83 HTR2C (0.42) HTR2CSLC6A4SLC16A3SLC16A1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed