SCHEMBL3701276

SCHEMBL3701276

Cn1c(C(=O)N2CCNCC2)cc2cc(Oc3ccc(NS(=O)(=O)c4ccc(C(F)(F)F)cc4)cn3)ccc21

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 19/20 0.51
SCN7A Q01118 6/20 0.51
KCNH2 Q12809 6/20 0.51
SCN10A Q9Y5Y9 3/20 0.51
SCN5A Q14524 1/20 0.51
SCN2A Q99250 1/20 0.51
SCN8A Q9UQD0 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3065606 0.97 SCN9A (0.49) SCN9ASCN7AKCNH2SCN10ASCN5A
Hydrochloric Acid SCHEMBL10180648 0.93 SCN9A (0.51) SCN9ASCN7AKCNH2SCN10ASCN5A
SCHEMBL3069830 0.89 SCN9A (0.47) SCN9A
Trifluoroacetic Acid SCHEMBL3061711 0.87 SCN9A (0.41) SCN9ASCN7AKCNH2SCN10ASCN5A
SCHEMBL3051748 0.87 SCN9A (0.53) SCN9ASCN7AKCNH2SCN10ASCN5A
SCHEMBL3064269 0.87 STAT3 (0.52) SCN9A
SCHEMBL3050791 0.86 SCN9A (0.51) SCN9ASCN10A
Hydrochloric Acid SCHEMBL3066788 0.86 SCN9A (0.49) SCN9ASCN7AKCNH2SCN10ASCN5A
Hydrochloric Acid SCHEMBL3053398 0.84 SCN9A (0.52) SCN9ASCN7AKCNH2SCN10ASCN5A
SCHEMBL3058988 0.83 STAT3 (0.49) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2207773-A2 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF Otsuka Pharmaceutical Co., Ltd. (JP) 2010-07-21 EP disclosed
WO-2009057811-A2 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2009-05-07 WO disclosed