SCHEMBL370163

SCHEMBL370163

Cc1ccccc1C(C/C(=N/O)c1ccc(=O)n(C)c1)c1ccc([C@H]2CC[C@@H](C(=O)O)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 7/20 0.51
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
APAF1 O14727 1/20 0.35
BRD4 O60885 1/20 0.33
FFAR1 O14842 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C1 Q04828 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
S1PR5 Q9H228 1/20 0.31
SLC6A1 P30531 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1390235 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL1389850 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL1390613 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL370165 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL1390234 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL370166 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL1389856 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL1390568 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL1389852 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4
SCHEMBL1390567 1.00 GPBAR1 (0.51) GPBAR1NPC1RAB9AAPAF1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed