SCHEMBL370209

SCHEMBL370209

Cc1cc(/C(CC(c2cccc(CC(=O)O)c2)c2ccccc2C)=N/O)ccn1.Cc1cc(C(CC(c2cccc(-c3ccc(S(C)(=O)=O)cc3)c2)c2ccccc2C)=NO)ccn1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 5/20 0.61
CTSA P10619 4/20 0.36
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
WNT3A P56704 4/20 0.34
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1389741 0.93 GPBAR1 (0.67) GPBAR1CTSAPSEN1PSEN2APH1B
SCHEMBL10241016 0.93 GPBAR1 (0.67) GPBAR1CTSAPSEN1PSEN2APH1B
SCHEMBL1389740 0.93 GPBAR1 (0.67) GPBAR1CTSAPSEN1PSEN2APH1B
SCHEMBL1389913 0.89 GPBAR1 (0.67) GPBAR1CTSA
SCHEMBL365003 0.89 GPBAR1 (0.67) GPBAR1CTSA
SCHEMBL363141 0.84 GPBAR1 (0.54) GPBAR1CTSACTSSCTSK
SCHEMBL10240885 0.84 GPBAR1 (0.54) GPBAR1CTSACTSSCTSK
SCHEMBL363140 0.84 GPBAR1 (0.54) GPBAR1CTSACTSSCTSK
SCHEMBL1390079 0.84 GPBAR1 (0.53) GPBAR1CTSAPSEN1PSEN2APH1B
SCHEMBL363578 0.84 GPBAR1 (0.86) GPBAR1CTSAPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2593426-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F.HOFFMANN-LA ROCHE AG (CH) 2013-05-22 EP disclosed
WO-2012007365-A1 1-HYDROXYIMINO-3-PHENYL-PROPANES F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed