SCHEMBL3704205

SCHEMBL3704205

Cc1cccc(Cn2cncc2CCN(C(=O)O)C(CC(C)C)C(=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 9/20 0.42
CYP11B2 P19099 9/20 0.42
ACE2 Q9BYF1 4/20 0.41
ACE P12821 3/20 0.41
FNTA P49354 2/20 0.38
FNTB P49356 2/20 0.38
PGGT1B P53609 1/20 0.38
LNPEP Q9UIQ6 1/20 0.36
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7381299 0.91 CYP11B1 (0.43) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL7382789 0.90 ACE2 (0.46) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL3681437 0.90 ACE2 (0.48) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL3714337 0.90 CYP11B1 (0.41) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL3710371 0.90 CYP11B1 (0.41) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL3715181 0.88 ACE2 (0.43) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL3712509 0.88 ACE2 (0.41) CYP11B1CYP11B2ACE2ACE
SCHEMBL7230044 0.87 ACE2 (0.41) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL7384484 0.87 CYP11B1 (0.41) CYP11B1CYP11B2ACE2ACEFNTA
SCHEMBL1655465 0.85 ACE2 (0.45) CYP11B1CYP11B2ACE2ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000066104-A9 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF MILLENNIUM PHARM INC (US) 2002-08-29 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2010093804-A1 ACE2 INHIBITORS FOR REDUCING GASTROINTESTINAL ADVERSE EFFECTS OF CYTOTOXIC AGENTS ORE PHARMACEUTICALS, INC. (US) 2010-08-19 WO disclosed
EP-1183019-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF Millennium Pharmaceuticals, Inc. (US) 2002-03-06 EP disclosed
WO-2000066104-A2 ACE-2 INHIBITING COMPOUNDS AND METHODS OF USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2000-11-09 WO disclosed