SCHEMBL3706282

SCHEMBL3706282

CSc1nc2nc(Cl)c(-c3ccccc3)cn2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.50
AKT1 P31749 6/20 0.44
AKT2 P31751 6/20 0.44
KDM4E B2RXH2 10/20 0.44
HPGD P15428 6/20 0.44
HSD17B10 Q99714 3/20 0.44
MAPT P10636 4/20 0.43
NPSR1 Q6W5P4 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
POLB P06746 1/20 0.43
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.39
PKM P14618 1/20 0.39
TSHR P16473 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
HTT P42858 2/20 0.39
CTDSP1 Q9GZU7 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL361914 0.82 KDM4E (0.46) ALDH1A1AKT1AKT2KDM4EHPGD
SCHEMBL362526 0.78 KMT2A (0.40) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL8012335 0.78 MAP4K4 (0.55) ALDH1A1KDM4EHPGDHSD17B10MAPT
SCHEMBL2967067 0.77 AKT1 (0.45) ALDH1A1AKT1AKT2KDM4EHPGD
SCHEMBL2968149 0.77 HPGD (0.41) ALDH1A1AKT1AKT2KDM4EHPGD
SCHEMBL3702122 0.76 AKT1 (0.54) ALDH1A1AKT1AKT2KDM4EHPGD
SCHEMBL3702899 0.75 AKT1 (0.47) ALDH1A1AKT1AKT2KDM4EHPGD
SCHEMBL867493 0.71 AKT1 (0.56) AKT1AKT2
SCHEMBL867191 0.70 SRC (0.39) ALDH1A1KDM4EHPGDMAPTSMN1; SMN2
SCHEMBL3707392 0.69 AKT1 (0.45) ALDH1A1AKT1AKT2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2396330-A1 FUSED PYRIMIDINES Bayer Pharma Aktiengesellschaft (DE) 2011-12-21 EP disclosed
WO-2010091808-A1 FUSED PYRIMIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-08-19 WO disclosed