SCHEMBL3708466

SCHEMBL3708466

C[C@@H]1CN(Cc2ccccn2)CCN1C(=O)c1cc2cc(Oc3ccc(N(C)C(=O)c4ccc(C(F)(F)F)cc4)cn3)ccc2n1C

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 7/20 0.49
MGLL Q99685 2/20 0.44
MLNR O43193 4/20 0.40
STAT3 P40763 4/20 0.39
CHRM4 P08173 1/20 0.38
PIK3CA P42336 1/20 0.38
PRKAA2 P54646 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10181162 1.00 SCN9A (0.49) SCN9AMGLLMLNRSTAT3CHRM4
SCHEMBL10181164 1.00 SCN9A (0.49) SCN9AMGLLMLNRSTAT3CHRM4
SCHEMBL3050999 0.93 MLNR (0.46) SCN9AMGLLMLNR
SCHEMBL3066677 0.91 SCN9A (0.59) SCN9ASTAT3PIK3CAPRKAA2
SCHEMBL3064516 0.89 SCN9A (0.49) SCN9AMGLLSTAT3
SCHEMBL3064521 0.89 SCN9A (0.49) SCN9AMGLLSTAT3
SCHEMBL3067772 0.89 SCN9A (0.49) SCN9AMGLLSTAT3
Oxalic Acid SCHEMBL3056958 0.87 STAT3 (0.48) MGLLMLNRSTAT3PIK3CAPRKAA2
Oxalic Acid SCHEMBL3064025 0.87 STAT3 (0.48) MGLLMLNRSTAT3PIK3CAPRKAA2
Oxalic Acid SCHEMBL10181285 0.87 STAT3 (0.48) MGLLMLNRSTAT3PIK3CAPRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2207773-B1 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF OTSUKA PHARMA CO LTD (JP) 2012-07-11 EP disclosed
EP-2207773-A2 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF Otsuka Pharmaceutical Co., Ltd. (JP) 2010-07-21 EP disclosed
WO-2009057811-A2 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2009-05-07 WO disclosed