SCHEMBL3709833

SCHEMBL3709833

Nc1cc2c(cc1N)C(O)CN(C(=O)C(F)(F)F)CC2.[Pd]

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 9/20 0.42
ESR2 Q92731 9/20 0.42
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
DRD1 P21728 2/20 0.33
PKM P14618 1/20 0.32
MTNR1B P49286 1/20 0.32
GRIN1 Q05586 2/20 0.32
GRIN2B Q13224 2/20 0.32
ABHD6 Q9BV23 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Water SCHEMBL3709828 0.80 ESR1 (0.54) ESR1ESR2CA12CA1CA2
SCHEMBL719456 0.80 ESR1 (0.56) ESR1ESR2CA12CA1CA2
Water SCHEMBL3709830 0.77 ESR1 (0.57) ESR1ESR2CA12CA1CA2
SCHEMBL4663870 0.77 GRIN1 (0.48) ESR1ESR2GRIN1GRIN2BABHD6
SCHEMBL25204719 0.70 ESR1 (0.53) ESR1ESR2PKMABHD6
SCHEMBL30411738 0.70 ESR1 (0.53) ESR1ESR2PKMABHD6
SCHEMBL25205929 0.70 ESR1 (0.53) ESR1ESR2PKMABHD6
SCHEMBL6395748 0.70 ESR1 (0.37) ESR1ESR2
SCHEMBL13561414 0.70 ESR1 (0.37) ESR1ESR2
SCHEMBL225186 0.70 ESR1 (0.37) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096384-A2 FUSED BENZAZEPINES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS TARGACEPT, INC. (US) 2010-08-26 WO disclosed