SCHEMBL3712243

SCHEMBL3712243

O=C(NO)c1c[c]nc(-c2ccc(C#Cc3cccnc3)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 10/20 0.45
HDAC1 Q13547 7/20 0.45
FFAR1 O14842 1/20 0.42
KDM1A O60341 1/20 0.40
SMPD1 P17405 1/20 0.40
HIF1A Q16665 1/20 0.39
EPAS1 Q99814 1/20 0.39
HDAC2 Q92769 5/20 0.38
HDAC8 Q9BY41 4/20 0.38
HDAC3 O15379 4/20 0.38
CSF1R P07333 1/20 0.37
CYP2A6 P11509 1/20 0.36
CYP2C9 P11712 1/20 0.36
CHRNB2 P17787 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
CHRNA4 P43681 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HDAC4 P56524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714897 0.84 HDAC1 (0.52) HDAC6HDAC1FFAR1KDM1ASMPD1
SCHEMBL3713444 0.81 HDAC6 (0.44) HDAC6HDAC1FFAR1KDM1ASMPD1
SCHEMBL13188328 0.80 HDAC6 (0.51) HDAC6HDAC1FFAR1KDM1AHIF1A
SCHEMBL400670 0.80 HDAC1 (0.60) HDAC6HDAC1FFAR1KDM1AHIF1A
SCHEMBL13188263 0.79 HDAC6 (0.42) HDAC6HDAC1FFAR1KDM1AHIF1A
SCHEMBL3713649 0.79 HDAC1 (0.52) HDAC6HDAC1FFAR1KDM1ASMPD1
SCHEMBL13188441 0.78 CSF1R (0.43) HDAC6HDAC1FFAR1KDM1ASMPD1
SCHEMBL3714241 0.78 HDAC6 (0.41) HDAC6HDAC1FFAR1KDM1AHIF1A
SCHEMBL3721790 0.78 HDAC6 (0.41) HDAC6HDAC1FFAR1KDM1AHIF1A
SCHEMBL3803200 0.78 ALDH2 (0.42) HDAC6HDAC1FFAR1KDM1AHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed