SCHEMBL3712915

SCHEMBL3712915

CCn1cnc2c(NCc3cccc(OC)c3N)nc(NCC(C)(O)C(C)C)nc21

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 12/20 0.51
CDK2 P24941 12/20 0.51
CCNT1 O60563 5/20 0.51
CDK9 P50750 5/20 0.51
CDK5 Q00535 5/20 0.51
CDK5R1 Q15078 5/20 0.51
CDK7 P50613 3/20 0.51
CCNH P51946 3/20 0.51
CDK1 P06493 5/20 0.45
CCNT2 O60583 2/20 0.45
CCNE2 O96020 2/20 0.45
PRKCA P17252 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1354863 0.92 CCNE1 (0.56) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1352736 0.89 CCNE1 (0.47) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1355210 0.88 CCNE1 (0.51) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1355393 0.88 CDK2 (0.51) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1354660 0.87 CCNE1 (0.57) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1355229 0.86 CDK2 (0.49) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1354680 0.85 CDK2 (0.53) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1354202 0.83 CDK1 (0.56) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1355081 0.83 CDK2 (0.54) CCNE1CDK2CCNT1CDK9CDK5
SCHEMBL1353769 0.82 CDK2 (0.75) CCNE1CDK2CCNT1CDK9CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391626-A2 SUBSTITUTED 6-(2-AMINOBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND PREPARATIONS CONTAINING THESE COMPOUNDS Univerzita Palackého v Olomouci (CZ) 2011-12-07 EP disclosed
WO-2010085924-A2 SUBSTITUTED 6-(2-AMINOBENZYLAMINO)PURINE DERIVATIVES, THEIR USE AS MEDICAMENTS AND PREPARATIONS CONTAINING THESE COMPOUNDS UNIVERZITA PALACKEHO V OLOMOUCI (CZ) 2010-08-05 WO disclosed