SCHEMBL3714522

SCHEMBL3714522

CC(=O)Nc1cccc(Nc2nccc(Nc3ccc(N)cc3)n2)c1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AURKA O14965 4/20 0.66
AURKB Q96GD4 2/20 0.66
SRC P12931 1/20 0.59
ITK Q08881 1/20 0.57
PLK1 P53350 1/20 0.56
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
JAK2 O60674 3/20 0.54
SYK P43405 2/20 0.54
JAK3 P52333 1/20 0.53
MAP3K5 Q99683 1/20 0.53
KIT P10721 1/20 0.52
FLT3 P36888 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27075730 0.89 PLK1 (0.70) AURKAAURKBSRCITKPLK1
SCHEMBL27075736 0.87 AURKA (0.73) AURKAAURKBSRCITKPLK1
SCHEMBL27075726 0.86 NPC1 (0.67) AURKAAURKBSRCITKPLK1
SCHEMBL27075735 0.85 AURKA (0.66) AURKAAURKBSRCSYK
SCHEMBL27075738 0.84 TNNI3K (0.62) AURKAAURKBSRCITKPLK1
SCHEMBL27075737 0.83 BRAF (0.60) AURKAAURKBSRCITKPLK1
SCHEMBL12968974 0.83 ROCK1 (0.66) AURKAAURKBSRCITKRAB9A
Hydrochloric Acid SCHEMBL12813262 0.82 ROCK1 (0.64) AURKAAURKBSRCITKRAB9A
SCHEMBL18780746 0.81 AURKA (0.54) AURKAAURKBNPC1RAB9ASYK
SCHEMBL27075734 0.80 AURKA (0.56) AURKAAURKBSRCITKPLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129802-A1 INHIBITORS OF JAK PORTOLA PHARMACEUTICALS, INC. (US) 2010-11-11 WO claimed