SCHEMBL3715089

SCHEMBL3715089

CN(C)Cc1cccc(C#Cc2ccc(-c3cc(C(=O)NO)ccn3)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 14/20 0.48
KDM1A O60341 10/20 0.48
EGFR P00533 3/20 0.47
HDAC6 Q9UBN7 3/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
FFAR1 O14842 1/20 0.42
PTGES O14684 1/20 0.41
AKR1C3 P42330 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3713122 0.88 KDM5B (0.45) EGFRFFAR1PTGESAKR1C3
SCHEMBL13187971 0.82 HDAC1 (0.61) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL13187738 0.82 HDAC1 (0.55) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL13188523 0.79 HDAC1 (0.55) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL3721374 0.78 FFAR1 (0.48) HDAC1KDM1AFFAR1
SCHEMBL3713063 0.78 HDAC1 (0.66) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL3714564 0.78 KDM4E (0.49) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL3714897 0.77 HDAC1 (0.52) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL13187716 0.73 HDAC1 (0.55) HDAC1KDM1AHDAC6HDAC2HDAC8
SCHEMBL13187834 0.73 HDAC6 (0.42) HDAC1HDAC6HDAC2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed
WO-2010100475-A1 HYDROXAMIC ACID DERIVATIVES AS GRAM-NEGATIVE ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2010-09-10 WO disclosed