SCHEMBL3715090

SCHEMBL3715090

O=C(c1ccc(-c2ncc[nH]2)cc1)N1CCCCCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.59
KDM4E B2RXH2 2/20 0.59
HPGD P15428 7/20 0.57
MAPK1 P28482 1/20 0.53
HTR2B P41595 4/20 0.52
RIPK1 Q13546 2/20 0.51
PDE4A P27815 1/20 0.49
PDE4B Q07343 1/20 0.49
PDE4C Q08493 1/20 0.49
PDE4D Q08499 1/20 0.49
KCNH2 Q12809 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
TSHR P16473 2/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CA12 O43570 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15154800 0.79 GAA (0.59) ALDH1A1KDM4EHPGDHTR2BPDE4A
SCHEMBL17303458 0.76 KDM4E (0.77) ALDH1A1KDM4EPDE4APDE4BPDE4C
SCHEMBL27479149 0.76 HPGD (1.00) ALDH1A1HPGDMAPK1TSHRMEN1
SCHEMBL7132525 0.76 HPGD (1.00) ALDH1A1HPGDMAPK1TSHRMEN1
SCHEMBL1060312 0.75 KDM4E (1.00) ALDH1A1KDM4EHPGDPDE4APDE4B
SCHEMBL8947386 0.74 HPGD (0.57) ALDH1A1HPGDMAPK1RIPK1TSHR
SCHEMBL857458 0.74 IKBKB (0.63) ALDH1A1HPGDRIPK1GSK3AGSK3B
SCHEMBL10721733 0.74 HPGD (0.95) ALDH1A1KDM4EHPGDMAPK1TSHR
SCHEMBL7383120 0.73 KDM4E (0.72) ALDH1A1KDM4EPDE4APDE4BPDE4C
SCHEMBL2424622 0.73 HTT (0.49) ALDH1A1HPGDHTR2BRIPK1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2391625-A1 NEW ADENOSINE RECEPTOR LIGANDS AND USES THEREOF Domain Therapeutics (FR) 2011-12-07 EP disclosed
WO-2010084425-A1 NEW ADENOSINE RECEPTOR LIGANDS AND USES THEREOF DOMAIN THERAPEUTICS (FR) 2010-07-29 WO disclosed