SCHEMBL3716072

SCHEMBL3716072

Nc1cc(F)c(F)c(C=O)c1F

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA7 P43166 2/20 0.37
CA13 Q8N1Q1 1/20 0.37
CA4 P22748 1/20 0.32
CA6 P23280 1/20 0.32
CA5A P35218 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
CA5B Q9Y2D0 1/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 1/20 0.32
KMT2A Q03164 1/20 0.32
CES2 O00748 2/20 0.31
CES1 P23141 2/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL441131 0.83 CA1 (0.44) CA12CA1CA2CA7CA13
SCHEMBL2562870 0.82 CA12 (0.37) CA12CA1CA2CA7CA13
SCHEMBL8684580 0.77 CA1 (0.41) CA12CA1CA2CA7CA13
SCHEMBL18526977 0.73 ERN1 (0.38) CA12CA1CA2CA7CA13
SCHEMBL9478821 0.73 CA1 (0.37) CA12CA1CA2CA7CA13
SCHEMBL4746715 0.73 ERN1 (0.35) CA12CA1CA2CA7CA13
SCHEMBL31015984 0.73 CA1 (0.37) CA12CA1CA2CA7CA13
SCHEMBL2891346 0.73 CYP2C9 (0.41) CA12CA1CA2CA7CA4
SCHEMBL19126540 0.73 CA12 (0.36) CA12CA1CA2CA7CA4
SCHEMBL17541205 0.72 CA1 (0.44) CA12CA1CA2CA7CA13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7858349-B2 Anti-cancer compounds THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2010-12-28 US disclosed
WO-2010127381-A1 DIAGNOSIS, MONITORING, PROGNOSIS, PREVENTION AND TREATMENT OF ANEURYSMS JAMES COOK UNIVERSITY (AU) 2010-11-11 WO disclosed
US-20090088454-A1 ANTI-CANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2009-04-02 US disclosed
US-7427496-B2 Anti-cancer compounds THE REGENTS OF THE UNIVERSITY OF COLORADO (US) 2008-09-23 US disclosed
US-20060183772-A1 To inhibit tumor growth in an animal; to induce apoptosis NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2006-08-17 US disclosed