SCHEMBL3716239

SCHEMBL3716239

CC(C)CC1c2cccc(-c3noc(-c4ccc(OC(C)C)c(Cl)c4)n3)c2CCN1C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.65
S1PR3 Q99500 6/20 0.65
CYP2C9 P11712 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3664014 0.95 S1PR1 (0.63) S1PR1S1PR3
SCHEMBL2124895 0.92 S1PR1 (0.58) S1PR1S1PR3CYP2C9
SCHEMBL2125906 0.90 S1PR1 (0.67) S1PR1S1PR3
SCHEMBL3664817 0.88 S1PR1 (0.63) S1PR1S1PR3
SCHEMBL3716238 0.87 S1PR1 (0.64) S1PR1S1PR3
SCHEMBL3664011 0.83 S1PR1 (0.62) S1PR1S1PR3
SCHEMBL2123484 0.81 S1PR1 (0.63) S1PR1S1PR3CYP2C9
SCHEMBL3664816 0.81 S1PR1 (0.62) S1PR1S1PR3
SCHEMBL2125344 0.81 S1PR1 (0.53) S1PR1S1PR3
SCHEMBL10130678 0.79 S1PR1 (0.77) S1PR1S1PR3CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225233-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (S1P) Glaxo Group Limited (GB) 2010-09-08 EP disclosed
EP-2222671-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (SIP) Glaxo Group Limited (GB) 2010-09-01 EP disclosed
WO-2009080724-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (S1P) GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed
WO-2009080728-A1 OXADIAZOLE DERIVATIVES ACTIVE ON SPHINGOSINE-1-PHOSPHATE (SIP) GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed