SCHEMBL3718302

SCHEMBL3718302

CC(C)(C)OC(=O)N1CCc2cc3nccnc3cc2CC1.c1cnc2cc3c(cc2n1)CCNCC3

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.49
NR1H2 P55055 1/20 0.45
GPR119 Q8TDV5 4/20 0.43
MAPK1 P28482 1/20 0.43
POLB P06746 1/20 0.41
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.40
THRB P10828 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
GRM5 P41594 1/20 0.39
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
FAAH O00519 1/20 0.39
HTT P42858 1/20 0.39
USP2 O75604 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7082357 0.78 ESR2 (0.53) ESR2NR1H2GPR119MAPK1NPC1
SCHEMBL7082361 0.77 NR1H2 (0.54) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL719713 0.74 NR1H2 (0.62) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL1294417 0.73 ESR2 (0.50) ESR2NR1H2GPR119MAPK1POLB
SCHEMBL5458949 0.72 ESR2 (0.52) ESR2NR1H2GPR119MAPK1MAPT
SCHEMBL2313024 0.72 ESR2 (0.48) ESR2NR1H2GPR119MAPTKDM4E
SCHEMBL2312041 0.72 ESR2 (0.48) ESR2NR1H2GPR119MAPTNPC1
SCHEMBL1225127 0.71 USP2 (0.58) NR1H2GPR119MAPK1MAPTKDM4E
SCHEMBL587550 0.71 USP2 (0.58) NR1H2GPR119MAPK1MAPTKDM4E
SCHEMBL8286 0.71 USP2 (0.58) NR1H2GPR119MAPK1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096384-A2 FUSED BENZAZEPINES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS TARGACEPT, INC. (US) 2010-08-26 WO disclosed