SCHEMBL3719147

SCHEMBL3719147

FC(F)(F)c1ccc(C2CCNCC2)cc1C(F)(F)F

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 10/20 0.61
QDPR P09417 1/20 0.51
HTR2A P28223 1/20 0.48
SLC18A3 Q16572 1/20 0.46
SIGMAR1 Q99720 1/20 0.46
PTPN5 P54829 1/20 0.42
SOS1 Q07889 1/20 0.41
CACNA1H O95180 1/20 0.39
TLR9 Q9NR96 2/20 0.39
TLR8 Q9NR97 2/20 0.39
TLR7 Q9NYK1 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5537443 0.86 HTR2C (0.57) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL4949183 0.86 HTR2C (0.57) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL5584686 0.85 HTR2C (0.56) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL30228395 0.85 HTR2C (0.56) HTR2CQDPRHTR2ASLC18A3SIGMAR1
Hydrochloric Acid SCHEMBL4893701 0.85 HTR2C (0.58) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL31342813 0.85 HTR2C (0.56) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL29623419 0.85 HTR2C (0.56) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL2710169 0.85 HTR2C (0.56) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL17102301 0.85 HTR2C (0.56) HTR2CQDPRHTR2ASLC18A3SIGMAR1
SCHEMBL30228726 0.85 HTR2C (0.56) HTR2CQDPRHTR2ASLC18A3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398796-A1 HETEROCYCLIC DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Canada Inc. (CA) 2011-12-28 EP disclosed
WO-2010094126-A1 HETEROCYCLIC DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2010-08-26 WO disclosed