SCHEMBL3719477

SCHEMBL3719477

CC1=C(C(N)=O)C(c2ccc(C#N)cc2S(C)(=O)=O)NC(=O)N1c1cccc(C(F)(F)F)c1

nearest known ligand 0.86

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ELANE P08246 20/20 0.86
CYP2C19 P33261 1/20 0.67
CYP2C9 P11712 3/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL122597 1.00 ELANE (0.86) ELANECYP2C19CYP2C9
SCHEMBL125346 0.92 ELANE (1.00) ELANECYP2C19CYP2C9
SCHEMBL18086937 0.92 ELANE (0.87) ELANECYP2C19CYP2C9
SCHEMBL123843 0.92 ELANE (1.00) ELANECYP2C19CYP2C9
SCHEMBL122465 0.92 ELANE (0.87) ELANECYP2C19CYP2C9
SCHEMBL123537 0.92 ELANE (0.87) ELANECYP2C19CYP2C9
SCHEMBL121576 0.92 ELANE (0.72) ELANECYP2C19CYP2C9
SCHEMBL123028 0.91 ELANE (0.71) ELANECYP2C19CYP2C9
SCHEMBL124616 0.90 ELANE (0.70) ELANECYP2C19CYP2C9
SCHEMBL125599 0.90 ELANE (0.76) ELANECYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234985-A1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF Bayer Schering Pharma Aktiengesellschaft (DE) 2010-10-06 EP disclosed
WO-2009080199-A1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed