SCHEMBL3720105

SCHEMBL3720105

CC(C)c1n[nH]c2c(NCc3cccc(F)c3)nc(NCC(O)CN)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.44
CDK9 P50750 2/20 0.44
CCNT1 O60563 1/20 0.43
PAK4 O96013 2/20 0.39
PLK4 O00444 1/20 0.39
CCNE1 P24864 4/20 0.39
CDK5 Q00535 3/20 0.39
APP P05067 2/20 0.37
NTRK1 P04629 5/20 0.37
CDK1 P06493 3/20 0.36
CDK7 P50613 2/20 0.36
AURKA O14965 3/20 0.36
AURKB Q96GD4 2/20 0.36
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
ABL1 P00519 1/20 0.36
LCK P06239 1/20 0.36
CSF1R P07333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722170 0.86 CCNE1 (0.44) CDK2CDK9CCNT1PLK4CCNE1
SCHEMBL3724956 0.85 CDK2 (0.42) CDK2CDK9CCNT1PAK4PLK4
SCHEMBL3720099 0.84 CDK2 (0.56) CDK2CDK9CCNT1CCNE1CDK5
SCHEMBL3717714 0.83 CDK2 (0.42) CDK2CDK9PAK4PLK4CCNE1
SCHEMBL3794940 0.80 CDK2 (0.35) CDK2CDK9CCNE1CDK5CDK1
SCHEMBL18396850 0.80 CDK2 (0.44) CDK2CDK9CCNT1CCNE1CDK5
SCHEMBL3721978 0.79 CCNE1 (0.42) CDK2CDK9CCNT1CCNE1CDK5
SCHEMBL3715540 0.79 CDK2 (0.57) CDK2CDK9CCNT1CCNE1CDK5
SCHEMBL3718107 0.77 CDK2 (0.59) CDK2CDK9CCNT1CCNE1CDK5
SCHEMBL2912272 0.76 CDK2 (0.51) CDK2CDK9CCNT1CCNE1CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010139288-A1 5,7-DISUBSTITUTED 3-ISOPROPYLPYRAZOLO[4,3-D]PYRIMIDINES FOR USE AS MEDICAMENTS AND PHARMACEUTICAL COMPOSITIONS C3 BIO GMBH (DE) 2010-12-09 WO disclosed