SCHEMBL3720239

SCHEMBL3720239

N#Cc1cccc(-c2cc(C(N)=O)nc(N3CCN(c4ccccc4F)CC3)n2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.54
HTT P42858 2/20 0.54
GLA P06280 1/20 0.54
ALDH1A1 P00352 4/20 0.53
HSD17B10 Q99714 3/20 0.53
GAA P10253 2/20 0.53
HPGD P15428 2/20 0.53
TSHR P16473 1/20 0.53
CASP1 P29466 1/20 0.53
CASP7 P55210 1/20 0.53
LMNA P02545 1/20 0.52
POLB P06746 1/20 0.52
GPR55 Q9Y2T6 1/20 0.52
HRH4 Q9H3N8 1/20 0.45
MAPK1 P28482 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
USP2 O75604 1/20 0.43
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3727226 0.90 KDM4E (0.56) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3721775 0.87 KDM4E (0.59) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3718588 0.87 KDM4E (0.71) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3726351 0.85 KDM4E (0.57) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL1733486 0.85 KDM4E (0.71) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3721015 0.83 KDM4E (0.55) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3720819 0.83 KDM4E (0.57) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3721046 0.83 KDM4E (0.58) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3727039 0.83 KDM4E (0.61) KDM4EHTTGLAALDH1A1HSD17B10
SCHEMBL3720242 0.82 HRH4 (0.46) KDM4EHTTALDH1A1LMNAHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed