SCHEMBL3721054

SCHEMBL3721054

c1nc(N2CCOCC2)nc2c1COCC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
HSP90AB1 P08238 2/20 0.47
ALDH1A1 P00352 3/20 0.46
POLB P06746 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
MAPK1 P28482 1/20 0.46
TSHR P16473 2/20 0.44
PIK3CA P42336 2/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CB P42338 1/20 0.43
HSP90AA1 P07900 1/20 0.43
KMT2A Q03164 2/20 0.43
ABL1 P00519 1/20 0.40
BCR P11274 1/20 0.40
PIK3R1 P27986 1/20 0.40
MTOR P42345 1/20 0.40
HPGD P15428 1/20 0.40
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13690044 0.84 HSP90AB1 (0.50) HSP90AB1ALDH1A1POLBSMN1; SMN2TSHR
SCHEMBL1364993 0.84 PTPN11 (0.39) KDM4EHSP90AB1ALDH1A1POLBSMN1; SMN2
SCHEMBL1366043 0.79 MKNK1 (0.40) HSP90AB1POLBSMN1; SMN2
SCHEMBL1020021 0.79 POLB (0.72) KDM4EHSP90AB1ALDH1A1POLBSMN1; SMN2
SCHEMBL24920531 0.78 HSP90AB1 (0.56) KDM4EHSP90AB1ALDH1A1POLBHSP90AA1
SCHEMBL12142170 0.76 HSP90AB1 (0.35) HSP90AB1ALDH1A1POLBSMN1; SMN2HSP90AA1
SCHEMBL12143536 0.76 HSP90AB1 (0.37) HSP90AB1ALDH1A1POLBSMN1; SMN2MAPK1
SCHEMBL17624125 0.75 HSP90AB1 (0.50) KDM4EHSP90AB1ALDH1A1POLBMAPK1
SCHEMBL2807505 0.75 POLB (0.56) KDM4EHSP90AB1ALDH1A1POLBSMN1; SMN2
SCHEMBL24921798 0.75 HSP90AB1 (0.47) KDM4EHSP90AB1ALDH1A1POLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120987-A1 RING FUSED, UREIDOARYL- AND CARBAMOYLARYL-BRIDGED MORPHOLINO-PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-10-21 WO disclosed