SCHEMBL3721732

SCHEMBL3721732

O=Cc1ccnc(-c2cnccn2)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
MAPT P10636 2/20 0.43
PIM2 Q9P1W9 2/20 0.40
PIM1 P11309 4/20 0.38
KDM1A O60341 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.36
CYP2A6 P11509 1/20 0.35
P2RX7 Q99572 1/20 0.34
TTK P33981 1/20 0.34
NISCH Q9Y2I1 1/20 0.33
CYP3A4 P08684 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
CCR1 P32246 1/20 0.33
CCR5 P51681 1/20 0.33
CCR8 P51685 1/20 0.33
ALOX5 P09917 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30796270 1.00 KDM4E (0.44) KDM4EMAPTPIM2PIM1KDM1A
SCHEMBL730405 0.86 CCR1 (0.42) KDM4ECYP2A6ALDH1A1CCR1CCR5
SCHEMBL29387096 0.86 CCR1 (0.42) KDM4ECYP2A6ALDH1A1CCR1CCR5
SCHEMBL30259554 0.84 CCR1 (0.41) KDM4EKDM1ACYP2A6ALDH1A1CCR1
SCHEMBL30259309 0.84 CCR1 (0.41) KDM4EKDM1ACYP2A6ALDH1A1CCR1
SCHEMBL19385092 0.79 CYP2A6 (0.60) PIM2PIM1KDM1AHDAC1HDAC6
SCHEMBL17057411 0.79 CYP2A6 (0.37) KDM4ECYP2A6ALDH1A1CCR1CCR5
SCHEMBL30541407 0.77 PIM2 (0.65) KDM4EMAPTPIM2PIM1TTK
SCHEMBL1313677 0.77 PIM2 (0.65) KDM4EMAPTPIM2PIM1TTK
SCHEMBL23787847 0.77 KDM4E (0.42) KDM4EKDM1AHDAC1HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010124055-A1 2-ALKYL PIPERIDINE MGLUR5 RECEPTOR MODULATORS MERCK SHARP & DOHME CORP. (US) 2010-10-28 WO claimed