SCHEMBL3721802

SCHEMBL3721802

Cc1n[nH]c(C)c1-c1cc(C(=O)c2nc3ccc(N4CCC(N(C)C)CC4)cc3[nH]2)ccn1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 6/20 0.76
CCND1 P24385 6/20 0.76
CCND3 P30281 5/20 0.70
CDK6 Q00534 5/20 0.70
CDK1 P06493 3/20 0.70
CCNB1 P14635 3/20 0.70
CCNA2 P20248 3/20 0.65
CDK2 P24941 3/20 0.65
CCNA1 P78396 3/20 0.65
FGFR1 P11362 2/20 0.38
PDGFRB P09619 1/20 0.38
KDR P35968 1/20 0.38
ATR Q13535 3/20 0.37
BRD4 O60885 3/20 0.36
FLT1 P17948 1/20 0.36
PDE10A Q9Y233 2/20 0.35
USP30 Q70CQ3 1/20 0.35
FLT3 P36888 1/20 0.35
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL110731 0.87 CDK4 (1.00) CDK4CCND1CCND3CDK6CDK1
SCHEMBL110695 0.86 CDK4 (0.73) CDK4CCND1CCND3CDK6CDK1
SCHEMBL112928 0.86 CDK4 (0.72) CDK4CCND1CCND3CDK6CDK1
SCHEMBL111515 0.86 CDK4 (0.57) CDK4CCND1CCND3CDK6CDK1
SCHEMBL2130180 0.85 CDK4 (0.58) CDK4CCND1CCND3CDK6CDK1
SCHEMBL109487 0.85 CDK4 (0.73) CDK4CCND1CCND3CDK6CDK1
SCHEMBL111810 0.84 CDK4 (0.83) CDK4CCND1CCND3CDK6CDK1
SCHEMBL112736 0.84 CDK4 (0.72) CDK4CCND1CCND3CDK6CDK1
SCHEMBL2129207 0.83 CDK4 (0.78) CDK4CCND1CCND3CDK6CDK1
SCHEMBL3722180 0.83 CDK4 (0.78) CDK4CCND1CCND3CDK6CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO claimed
WO-2010125402-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS MODULATORS OF CYCLIN DEPENDENT KINASES NOVARTIS AG (CH) 2010-11-04 WO disclosed