SCHEMBL3723767

SCHEMBL3723767

CCNc1cc(-c2ccc(NC(=O)NCc3ccc(N)nc3)c(F)c2)ccc1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 4/20 0.43
HDAC1 Q13547 3/20 0.42
MKNK1 Q9BUB5 1/20 0.38
MKNK2 Q9HBH9 1/20 0.38
CFD P00746 1/20 0.37
MAPK1 P28482 1/20 0.37
HPSE Q9Y251 2/20 0.36
RARB P10826 2/20 0.36
RARA P10276 1/20 0.36
RARG P13631 1/20 0.36
PDPK1 O15530 1/20 0.36
MTOR P42345 1/20 0.36
THRB P10828 1/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA5A P35218 1/20 0.35
CA9 Q16790 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3061231 0.88 NAMPT (0.53) NAMPTHDAC1MKNK1MKNK2
SCHEMBL3727393 0.85 NAMPT (0.42) NAMPTHDAC1MAPK1HPSEPDPK1
SCHEMBL485895 0.83 PIK3CA (0.44) NAMPTMTOR
SCHEMBL485974 0.81 HDAC1 (0.40) NAMPTHDAC1MAPK1PDPK1MTOR
SCHEMBL486537 0.79 ALOX5AP (0.41) NAMPTHDAC1MAPK1PDPK1MTOR
SCHEMBL485963 0.77 MTOR (0.45) NAMPTHDAC1MAPK1PDPK1MTOR
SCHEMBL486436 0.76 HDAC1 (0.37) NAMPTHDAC1MAPK1PDPK1MTOR
SCHEMBL3722076 0.76 HDAC1 (0.47) NAMPTHDAC1
SCHEMBL3719617 0.75 NAMPT (0.41) NAMPTHDAC1HPSEMTOR
SCHEMBL3048655 0.75 NAMPT (0.42) NAMPTMKNK1MKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010109122-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF AS ANTICANCER DRUGS SANOFI-AVENTIS (FR) 2010-09-30 WO claimed
WO-2010109122-A1 NICOTINAMIDE DERIVATIVES, PREPARATION THEREOF, AND THERAPEUTIC USE THEREOF AS ANTICANCER DRUGS SANOFI-AVENTIS (FR) 2010-09-30 WO disclosed