SCHEMBL3723940

SCHEMBL3723940

O=C(Nc1ccc(-c2nc3c(c(N4C5CCC4COC5)n2)CNC3)cc1)Nc1cccnc1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MTOR P42345 18/20 0.61
PIK3CA P42336 16/20 0.61
PIK3CG P48736 9/20 0.61
PIK3CD O00329 2/20 0.49
CYP2C8 P10632 1/20 0.48
PIK3CB P42338 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3718615 0.93 MTOR (0.61) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL3721937 0.93 MTOR (0.59) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL3722519 0.87 MTOR (0.62) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL3721559 0.86 MTOR (0.66) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL3722650 0.86 MTOR (0.61) MTORPIK3CAPIK3CGPIK3CD
SCHEMBL3723078 0.86 MTOR (0.56) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL628043 0.85 MTOR (0.68) MTORPIK3CAPIK3CGPIK3CDCYP2C8
SCHEMBL3721995 0.83 MTOR (0.70) MTORPIK3CAPIK3CGPIK3CD
SCHEMBL3728020 0.83 MTOR (0.66) MTORPIK3CAPIK3CGPIK3CD
SCHEMBL3720999 0.81 MTOR (0.57) MTORPIK3CAPIK3CGPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120996-A1 5,6,7,8-TETRAHYDROPYRIDO[3,4-D]PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-10-21 WO disclosed