SCHEMBL3723982

SCHEMBL3723982

Cc1cc(F)cc(C)c1-c1ccccc1COc1cccc2cnccc12

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 2/20 0.46
KCNA3 P22001 1/20 0.46
NR3C1 P04150 2/20 0.42
MCL1 Q07820 1/20 0.39
NR2F2 P24468 1/20 0.38
RAB9A P51151 1/20 0.38
SGMS2 Q8NHU3 3/20 0.38
PDE10A Q9Y233 1/20 0.37
ADRB2 P07550 1/20 0.37
ADRB1 P08588 1/20 0.37
ADRB3 P13945 1/20 0.37
CNR2 P34972 1/20 0.37
CACNA2D1 P54289 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723393 0.83 GPBAR1 (0.46) GPBAR1KCNA3NR3C1NR2F2RAB9A
SCHEMBL3716494 0.80 GPBAR1 (0.57) GPBAR1KCNA3MCL1RAB9ASGMS2
SCHEMBL13152509 0.79 KCNA3 (0.56) GPBAR1KCNA3MCL1NR2F2RAB9A
SCHEMBL3713000 0.77 GPBAR1 (0.45) GPBAR1KCNA3NR3C1NR2F2RAB9A
SCHEMBL3715454 0.76 KCNA3 (0.48) GPBAR1KCNA3NR3C1NR2F2RAB9A
SCHEMBL13152511 0.75 GPBAR1 (0.43) GPBAR1KCNA3NR3C1NR2F2RAB9A
SCHEMBL31364101 0.70 KCNA3 (0.65) GPBAR1KCNA3NR2F2RAB9A
SCHEMBL5445170 0.70 KCNA3 (0.65) GPBAR1KCNA3NR2F2RAB9A
SCHEMBL3721720 0.69 GPBAR1 (0.54) GPBAR1KCNA3NR3C1NR2F2RAB9A
SCHEMBL11144866 0.68 KCNA3 (0.61) KCNA3NR3C1NR2F2RAB9ACACNA2D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010117090-A1 NOVEL ISOQUINOLINYLOXYMETHYL HETEROARYL DERIVATIVES BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-10-14 WO claimed
WO-2010117090-A1 NOVEL ISOQUINOLINYLOXYMETHYL HETEROARYL DERIVATIVES BANYU PHARMACEUTICAL CO.,LTD. (JP) 2010-10-14 WO disclosed