SCHEMBL3724872

SCHEMBL3724872

Nc1cccc(-c2nc(Cl)cc(N3CCOCC3)n2)c1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ATR Q13535 1/20 0.60
MAPT P10636 3/20 0.58
CYP1A2 P05177 2/20 0.58
HTT P42858 1/20 0.58
CYP2D6 P10635 1/20 0.58
PIK3CA P42336 11/20 0.55
NPSR1 Q6W5P4 2/20 0.54
TSHR P16473 1/20 0.54
MAPK1 P28482 1/20 0.54
HSD17B10 Q99714 1/20 0.54
PIK3CG P48736 4/20 0.54
MTOR P42345 3/20 0.54
PIK3CD O00329 2/20 0.54
PIK3CB P42338 3/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3878007 0.87 HTT (0.61) MAPTCYP1A2HTTCYP2D6PIK3CA
SCHEMBL1029661 0.85 HTT (0.80) ATRMAPTCYP1A2HTTCYP2D6
SCHEMBL4139135 0.85 PIK3CA (0.74) MAPTCYP1A2HTTCYP2D6PIK3CA
SCHEMBL1263306 0.85 ATR (0.60) ATRMAPTHTTPIK3CANPSR1
SCHEMBL4934392 0.81 PIK3CA (0.66) MAPTHTTPIK3CANPSR1TSHR
SCHEMBL4128517 0.81 CYP1A2 (0.61) ATRMAPTCYP1A2HTTCYP2D6
SCHEMBL1309606 0.80 PIK3CA (0.68) ATRHTTPIK3CANPSR1PIK3CG
SCHEMBL1029078 0.80 PIK3CA (0.63) MAPTCYP1A2HTTCYP2D6PIK3CA
SCHEMBL1263031 0.80 MAPT (0.54) ATRMAPTCYP1A2HTTCYP2D6
SCHEMBL4604779 0.79 PIK3CA (0.63) ATRMAPTCYP1A2HTTPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120994-A2 UREIDOARYL-AND CARBAMOYLARYL-MORPHOLINO- PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESIS WYETH LLC (US) 2010-10-21 WO disclosed